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European Journal of Drug Metabolism and Pharmacokinetics

Ausgabe 1/2023

Inhalt (12 Artikel)

Systematic Review

Hepatic Transporters Alternations Associated with Non-alcoholic Fatty Liver Disease (NAFLD): A Systematic Review

Navid Omidkhoda, Simin zare, Sina Mahdiani, Sara Samadi, Fatemeh Akhlaghi, Amir Hooshang Mohammadpour

Original Research Article

Population Pharmacokinetics and Dosing Simulations of Intravenous Oxycodone for Perioperative Pain Relief in Adult Surgical Patients with Obesity

Sook Hui Chaw, Yoke Lin Lo, Li Ling Yeap, Didi Erwandi Bin Mohamad Haron, Ina Ismiarti Shariffuddin

Original Research Article

Effect of Carbidopa Dose on Levodopa Pharmacokinetics With and Without Catechol-O-Methyltransferase Inhibition in Healthy Subjects

Johanna Tuunainen, Noora Sjöstedt, Mikko Vahteristo, Juha Ellmén, Mikko Kuoppamäki, Juha Rouru, Marjo Yliperttula

Open Access Original Research Article

Pharmacokinetics and Safety of Vedolizumab Following Administration of a Single Intravenous Dose in Healthy Chinese Subjects

Ran Xie, Nan Zhao, Bo Jia, Xia Zhao, Yimin Cui, Hiroyuki Okamoto, Lili Yang, Alexander Prokopienko

Original Research Article

Therapeutic Drug Monitoring of Lacosamide in Chinese Pediatric Patients with Epilepsy: Efficacy and Factors Influencing the Plasma Concentration

Ting Zhao, Hong-jian Li, Hui-lan Zhang, Jing Yu, Jie Feng, Ting-ting Wang, Yan Sun, Lu-hai Yu

Open Access Original Research Article

Pharmacokinetic Interactions and Tolerability of Rosuvastatin and Ezetimibe: A Randomized, Phase 1, Crossover Study in Healthy Chinese Participants

Lu Wang, Yingcai Luan, Chuandong Jia, Xin Xie, Zihao Zhang, Xiaochuan Xie, Qian Wang, Chanyan Hu, Fang Xie, Mohamed Abdel-Moneim, Lionel Hovsepian, Zhihong Zhao, Na Yang, Jie Hou

Original Research Article

Preclinical and Clinical Pharmacokinetics and Bioavailability in Healthy Volunteers of a Novel Formulation of the Selective P2X3 Receptor Antagonist Eliapixant

Klaus Francke, Niladri Chattopadhyay, Stefan Klein, Antje Rottmann, Dennis Krickau, Jeroen van de Wetering, Christian Friedrich

Original Research Article

Population Pharmacokinetic Analysis for Model-Based Therapeutic Drug Monitoring of Tacrolimus in Chinese Han Heart Transplant Patients

Yu Cheng, Jiana Chen, Xiaojuan Lin, Hongqiang Qiu, Jinhua Zhang

Open Access Original Research Article

Population Pharmacokinetic–Pharmacodynamic Modeling and Probability of Target Attainment Analysis of Rocuronium and Sugammadex in Children Undergoing Surgery

Małgorzata Grześkowiak, Agnieszka Bienert, Paweł Wiczling, Mirosław Malec, Joanna Grzelak, Konrad Jarosz, Justyna Ber, Michał Książkiewicz, Jowita Rosada-Kurasińska, Edmund Grześkowiak, Alicja Bartkowska-Śniatkowska

Research Letter

Rapid Brain Distribution of Subcutaneously Administered Methamphetamine in Mice

Greg Gorman, Lori Coward, Michael D. Hambuchen

Open Access Correction

Correction to: Evaluating Islatravir Administered Via Microneedle Array Patch for Long-Acting HIV Pre-exposure Prophylaxis Using Physiologically Based Pharmacokinetic Modelling

Hannah Kinvig, Nicolas Cottura, Andrew Lloyd, Collrane Frivold, Jessica Mistilis, Courtney Jarrahian, Marco Siccardi