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European Journal of Drug Metabolism and Pharmacokinetics

Ausgabe 1/2021

Inhalt (13 Artikel)

Review Article

Clinical Pharmacokinetics and Pharmacodynamics of Anti-Tubercular Drugs in Pregnancy

Jennifer R. Shiu, Alan Min, Tony K. L. Kiang

Review Article

The Impact of Fasting on Major Metabolic Pathways of Macronutrients and Pharmacokinetics Steps of Drugs

Reza Karimi, Anita Cleven, Fawzy Elbarbry, Huy Hoang

Original Research Article

Physiologically Based Pharmacokinetic Modeling Approach to Identify the Drug–Drug Interaction Mechanism of Nifedipine and a Proton Pump Inhibitor, Omeprazole

Maxime Le Merdy, Ming-Liang Tan, Dajun Sun, Zhanglin Ni, Sue-Chih Lee, Andrew Babiskin, Liang Zhao

Open Access Original Research Article

Population Pharmacokinetics of Cariprazine and its Major Metabolites

Antonia Periclou, Luann Phillips, Parviz Ghahramani, Margit Kapás, Timothy Carrothers, Tatiana Khariton

Open Access Original Research Article

Comparison of the Pharmacokinetics of RIPK1 Inhibitor GSK2982772 in Healthy Western and Japanese Subjects

Debra J. Tompson, Carwyn Davies, Nicola E. Scott, Edward P. Cannons, Michalis Kostapanos, Annette S. Gross, Marcy Powell, Hiroko Ino, Ryutaro Shimamura, Hirofumi Ogura, Takashi Nagakubo, Harue Igarashi, Atsushi Nakano

Open Access Original Research Article

The Effect of Verapamil, a P-gp Inhibitor, on the Pharmacokinetics, Safety, and Tolerability of Omadacycline in Healthy Adults: A Phase I, Open-Label, Single-Sequence Study

Thomas L. Hunt, Evan Tzanis, Stephen Bai, Amy Manley, Surya Chitra, Paul C. McGovern

Original Research Article

Differences in Intestinal Metabolism of Ginseng Between Normal and Immunosuppressed Rats

Jin-Hao Zhu, Jin-Di Xu, Shan-Shan Zhou, Xiao-Ya Zhang, Jing Zhou, Ming Kong, Qian Mao, He Zhu, Song-Lin Li

Original Research Article

Impact of Human SULT1E1 Polymorphisms on the Sulfation of 17β-Estradiol, 4-Hydroxytamoxifen, and Diethylstilbestrol by SULT1E1 Allozymes

Amal A. El Daibani, Fatemah A. Alherz, Maryam S. Abunnaja, Ahsan F. Bairam, Mohammed I. Rasool, Katsuhisa Kurogi, Ming-Cheh Liu

Original Research Article

Pharmacokinetics of the Urokinase Receptor-Derived Peptide UPARANT After Single and Multiple Doses Administration in Rats

Michele Ciccone, Daniele D’Alonzo, Alfonsina Mariarosaria Cangiano, Maria De Fenza, Vincenzo Pavone, Angelo Mancinelli

Original Research Article

Rapalogues as hCES2A Inhibitors: In Vitro and In Silico Investigations

Cheng-Cheng Shi, Yun-Qing Song, Rong-Jing He, Xiao-Qing Guan, Li-Lin Song, Shi-Tong Chen, Meng-Ru Sun, Guang-Bo Ge, Li-Rong Zhang

Open Access Original Research Article

Effect of Kidney Function and Dialysis on the Pharmacokinetics and Pharmacodynamics of Roxadustat, an Oral Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitor

Dorien Groenendaal-van de Meent, Virginie Kerbusch, Rudiger Kaspera, Begona Barroso-Fernandez, Piergiorgio Galletti, Gernot K. Klein, Martin den Adel

Open Access Short Communication

Comparison of Two Analytical Methods for Busulfan Therapeutic Drug Monitoring

Simona De Gregori, Carmine Tinelli, Federica Manzoni, Antonella Bartoli