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Drugs in R&D

Ausgabe 2/2022

Inhalt (8 Artikel)

Open Access Review Article

Exebacase: A Novel Approach to the Treatment of Staphylococcal Infections

Matthew W. McCarthy

Open Access Original Research Article

Pharmacokinetics and Safety of Ferric Pyrophosphate Citrate in Chinese Subjects with and without Hemodialysis-Dependent Stage 5 Chronic Kidney Disease

Liangying Gan, Panpan Xie, Yan Tan, Gang Wei, Xiaojuan Yuan, Zhifei Lu, Raymond Pratt, Yongchun Zhou, Ai-Min Hui, Kexin Li, Yi Fang, Li Zuo

Open Access Original Research Article

First-in-Human Phase I Study of the Novel Injectable Calcimimetic Agent Upacicalcet in Healthy Adult Japanese Participants

Fumihiko Koiwa, Rie Yazawa, Masafumi Fukagawa, Daisuke Honda, Tadao Akizawa

Open Access Original Research Article

A Phase I, Open-label, Single-Dose Study to Evaluate the Pharmacokinetics, Safety, and Tolerability of AMG 986 in Healthy Japanese Subjects

Ashit Trivedi, Omar Mather, Silvia Vega, Shauna Hutton, Jennifer Hellawell, Edward Lee

Open Access Original Research Article

Evaluation of the Pharmacokinetics and Safety of AMG 986 Tablet and Capsule Formulations in Healthy Adult Subjects: A Phase I, Open-Label, Randomized Study

Ashit Trivedi, Y.-H. Kiang, Robert E. Saw, Guilong Charles Cheng, Omar Mather, Silvia Vega, Jennifer Hellawell, Edward Lee

Open Access Original Research Article

Hydroxychloroquine Blood Concentrations Can Be Clinically Relevant Also After Drug Discontinuation

Simona De Gregori, Francesco Falaschi, Alessia Ballesio, Alessandra Fusco, Elisa Cremonte, Roberta Canta, Umberto Sabatini, Mariadelfina Molinaro, Carlo Soffiantini, Alba Nardone, Alessandro Vicentini, Annalisa De Silvestri, Antonio Di Sabatino

Open Access Original Research Article

Preclinical and Toxicology Studies of BRD5529, a Selective Inhibitor of CARD9

Theodore J. Kottom, Kyle Schaefbauer, Eva M. Carmona, Eunhee S. Yi, Andrew H. Limper

Open Access Original Research Article

Evaluation of the Effect of Food on the Pharmacokinetics of SHR6390, An Oral CDK4/6 Inhibitor, in Healthy Volunteers

Yan-ping Liu, Ming-hui Hu, Ping-ping Lin, Ting Li, Shu-qin Liu, Yu-ya Wang, Shao-rong Li, Xiang-kun Li, Chen-jing Wang, Yu Cao