Ausgabe 1/2024
Inhalt (10 Artikel)
Neural Network Models for Predicting Solubility and Metabolism Class of Drugs in the Biopharmaceutics Drug Disposition Classification System (BDDCS)
Aryan Ashrafi, Kiarash Teimouri, Farnaz Aghazadeh, Ali Shayanfar
Distribution, Metabolism, and Excretion of Cenobamate in Adult, Fetal, Neonatal, and Lactating Rats
Jairam Palamanda, Kelli J. Glenn, Susan M. Melnick
Pharmacokinetics of 4-Hydroxybenzaldehyde in Normal and Cerebral Ischemia–Reperfusion Injury Rats Based on Microdialysis Technique
Chunping Xu, Jin Feng, Hang Sun, Mingli Yan, Qian Yang, Xiaonan Zhou, Jianguang Yang, Fangyan He, Qing Lin
Ticagrelor Steady-State Trough Concentration in Chinese Patients Undergoing Percutaneous Coronary Intervention
ShaoJun Zheng, Qiong Jie, NaiDong Chen, XiJing Chen, YuBing Zhu
Pharmacokinetics of Imatinib Mesylate and Development of Limited Sampling Strategies for Estimating the Area under the Concentration–Time Curve of Imatinib Mesylate in Palestinian Patients with Chronic Myeloid Leukemia
Deema Hilmi Adawi, Nadia Ben Fredj, Ahmad Al-barghouthi, Ichrack Dridi, Mustafa Lubada, Mohammad Manasra, Karim Aouam
Pharmacokinetic Parameters of Recombinant Human Cyclophilin A in Mice
Anastasiia Kalinina, Elena Grigorieva, Anna Smirnova, Dmitry Kazansky, Ludmila Khromykh
Mass Balance and Metabolic Pathways of Eliapixant, a P2X3 Receptor Antagonist, in Healthy Male Volunteers
Stefanie Reif, Marcus-Hillert Schultze-Mosgau, Anna Engelen, Isabel Piel, Karsten Denner, Ad Roffel, Renger Tiessen, Stefan Klein, Klaus Francke, Antje Rottmann
Development, Physicochemical Characteristics and Pharmacokinetics of a New Sustained-Release Bilayer Tablet Formulation of Tramadol with an Immediate-Release Component for Twice-Daily Administration
Naoki Ishitsubo, Shinji Oguro, Hirotoshi Shimahashi, Masato Kawanishi, Takeshi Adachi, Kenji Mitsuda, Nobuyuki Ishibashi
Evaluation of Hydroxychloroquine as a Perpetrator on Cytochrome P450 (CYP) 3A and CYP2D6 Activity with Microdosed Probe Drugs in Healthy Volunteers
Felicitas Stoll, Antje Blank, Gerd Mikus, David Czock, Johanna Weiss, Marleen J. Meyer-Tönnies, Katja S. Gümüs, Mladen Tzvetkov, Jürgen Burhenne, Walter E. Haefeli
Comparative Pharmacokinetic Study of Rhubarb Anthraquinones in Normal and Nonalcoholic Fatty Liver Disease Rats
Fang Zhang, Rui Wu, Yanfang Liu, Shu Dai, Xinyan Xue, Xiaohong Gong, Yunxia Li