Ausgabe 4/2014
Inhalt (13 Artikel)
The use of a prodrug approach to minimize potential CNS exposure of next generation quinoline methanols while maintaining efficacy in in vivo animal models
Jason C. Sousa, Erin Milner, Dustin Carroll, William McCalmont, Sean Gardner, Jay Moon, Jacob D. Johnson, Patricia Lee, Jennifer Auschwitz, Norma Roncal, Diana Caridha, Anchalee Tungteung, Qiang Zeng, Sean Reyes, Bryan Smith, Qigui Li, Michael P. Kozar, Victor Melendez, Geoffrey Dow
Pharmacokinetic evaluation of formulated levodopa methyl ester nasal delivery systems
Yeon Hong Lee, Kyung Hee Kim, In Kyung Yoon, Kyung Eun Lee, In Koo Chun, Jeong Yeon Rhie, Hye Sun Gwak
The influence of comedication on tacrolimus blood concentration in patients subjected to kidney transplantation: a retrospective study
Neven Vavic, Nemanja Rancic, Viktorija Dragojevic-Simic, Biljana Draskovic-Pavlovic, Dubravko Bokonjic, Ljiljana Ignjatovic, Momir Mikov
Pharmacokinetics and hepatic uptake of gliquidone affected by Huangqi injection
Fan Zhang, Yuhui Wei, Yan Zhou, Dan Wang, Liting Zhou, Jianping Zhang, Xinan Wu
A comparison of in vitro ADME properties and pharmacokinetics of azithromycin and selected 15-membered ring macrolides in rodents
Astrid Milić, Vlatka Bencetić Mihaljević, Jovica Ralić, Ana Bokulić, Danijela Nožinić, Branka Tavčar, Boris Mildner, Vesna Munić, Ivica Malnar, Jasna Padovan
Effect of silibinin on the pharmacokinetics of nitrendipine in rabbits
Swathi Voruganti, Shravan Kumar Yamsani, Madhusudan Rao Yamsani
In vitro–in vivo evaluation of in situ gelling and thermosensitive ketoprofen liquid suppositories
Işık Özgüney, Anita Kardhiqi, Gülbeyaz Yıldız, Gökhan Ertan
Inhibition of murine cardiomyocyte respiration by amine local anesthetics
Elhadi H. Aburawi, Abdul-Kader Souid
Quantitative subcellular study of transferrin receptor-targeted doxorubicin and its metabolite in human breast cancer cells
Jinhui Xu, Yuan Sheng, Feifei Xu, Ying Yu, Yun Chen
Effects of silymarin on the pharmacokinetics of atorvastatin in diabetic rats
Hassan Malekinejad, Shirin Rokhsartalab-Azar, Sepideh Hassani-Dizaj, Shahin Alizadeh-Fanalou, Aysa Rezabakhsh, Amir Amniattalab
Gender differences in pharmacokinetics of a combination tablet of niacin extended-release/simvastatin in healthy Chinese volunteers
Xiao-lin Wang, Man Liu, Man Yang, Ya-nan Zhang, Dan Zhang, Li-na Zhang, Jing Han, Hui-chen Liu
The evaluation method for antiplatelet effect of acetylsalicylic acid
Haruko Yokoyama, Takashi Mastumura, Shinji Soeda, Yuji Suzuki, Masayuki Watanabe, Emiko Kashiwakura, Takayuki Saso, Noriyuki Ikeda, Kentaro Tokuoka, Yasuhisa Kitagawa, Yasuhiko Yamada
The metabolism of trifluoperazine (TFP) exhibits atypical kinetic behavior in both human liver microsomes (HLMs) and monkey liver microsomes (MyLM)
Jin-Fang Xiao, Xiao-Jun Liu, Gao-Wang Liu, Xue-Ying Yang, Pan Xiao, Xiao-Min Hou, Hai-Tang Wang, Jian-Jun Tang, Ya-Ting Zhang, Chen Zhen, Hai-Hong Fang