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European Journal of Drug Metabolism and Pharmacokinetics

Ausgabe 4/2014

Inhalt (13 Artikel)

Original Paper

The use of a prodrug approach to minimize potential CNS exposure of next generation quinoline methanols while maintaining efficacy in in vivo animal models

Jason C. Sousa, Erin Milner, Dustin Carroll, William McCalmont, Sean Gardner, Jay Moon, Jacob D. Johnson, Patricia Lee, Jennifer Auschwitz, Norma Roncal, Diana Caridha, Anchalee Tungteung, Qiang Zeng, Sean Reyes, Bryan Smith, Qigui Li, Michael P. Kozar, Victor Melendez, Geoffrey Dow

Original Paper

Pharmacokinetic evaluation of formulated levodopa methyl ester nasal delivery systems

Yeon Hong Lee, Kyung Hee Kim, In Kyung Yoon, Kyung Eun Lee, In Koo Chun, Jeong Yeon Rhie, Hye Sun Gwak

Original Paper

The influence of comedication on tacrolimus blood concentration in patients subjected to kidney transplantation: a retrospective study

Neven Vavic, Nemanja Rancic, Viktorija Dragojevic-Simic, Biljana Draskovic-Pavlovic, Dubravko Bokonjic, Ljiljana Ignjatovic, Momir Mikov

Original Paper

Pharmacokinetics and hepatic uptake of gliquidone affected by Huangqi injection

Fan Zhang, Yuhui Wei, Yan Zhou, Dan Wang, Liting Zhou, Jianping Zhang, Xinan Wu

Original Paper

A comparison of in vitro ADME properties and pharmacokinetics of azithromycin and selected 15-membered ring macrolides in rodents

Astrid Milić, Vlatka Bencetić Mihaljević, Jovica Ralić, Ana Bokulić, Danijela Nožinić, Branka Tavčar, Boris Mildner, Vesna Munić, Ivica Malnar, Jasna Padovan

Original Paper

Effect of silibinin on the pharmacokinetics of nitrendipine in rabbits

Swathi Voruganti, Shravan Kumar Yamsani, Madhusudan Rao Yamsani

Original Paper

In vitro–in vivo evaluation of in situ gelling and thermosensitive ketoprofen liquid suppositories

Işık Özgüney, Anita Kardhiqi, Gülbeyaz Yıldız, Gökhan Ertan

Original Paper

Inhibition of murine cardiomyocyte respiration by amine local anesthetics

Elhadi H. Aburawi, Abdul-Kader Souid

Original Paper

Effects of silymarin on the pharmacokinetics of atorvastatin in diabetic rats

Hassan Malekinejad, Shirin Rokhsartalab-Azar, Sepideh Hassani-Dizaj, Shahin Alizadeh-Fanalou, Aysa Rezabakhsh, Amir Amniattalab

Original Paper

Gender differences in pharmacokinetics of a combination tablet of niacin extended-release/simvastatin in healthy Chinese volunteers

Xiao-lin Wang, Man Liu, Man Yang, Ya-nan Zhang, Dan Zhang, Li-na Zhang, Jing Han, Hui-chen Liu

Original Paper

The evaluation method for antiplatelet effect of acetylsalicylic acid

Haruko Yokoyama, Takashi Mastumura, Shinji Soeda, Yuji Suzuki, Masayuki Watanabe, Emiko Kashiwakura, Takayuki Saso, Noriyuki Ikeda, Kentaro Tokuoka, Yasuhisa Kitagawa, Yasuhiko Yamada

Short Communication

The metabolism of trifluoperazine (TFP) exhibits atypical kinetic behavior in both human liver microsomes (HLMs) and monkey liver microsomes (MyLM)

Jin-Fang Xiao, Xiao-Jun Liu, Gao-Wang Liu, Xue-Ying Yang, Pan Xiao, Xiao-Min Hou, Hai-Tang Wang, Jian-Jun Tang, Ya-Ting Zhang, Chen Zhen, Hai-Hong Fang