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European Journal of Drug Metabolism and Pharmacokinetics

Ausgabe 4/2018

Inhalt (12 Artikel)

Review Article

Pharmacology of Pimasertib, A Selective MEK1/2 Inhibitor

Nuggehally R. Srinivas

Review Article

Pharmacokinetic Properties of Saffron and its Active Components

Azar Hosseini, Bibi Marjan Razavi, Hossein Hosseinzadeh

Original Research Article

Effects of Human Sulfotransferase 2A1 Genetic Polymorphisms 3 on the Sulfation of Tibolone

Ethan Miller, Munaf H. Zalzala, Maryam S. Abunnaja, Katsuhisa Kurogi, Yoichi Sakakibara, Masahito Suiko, Ming-Cheh Liu

Original Research Article

Genotyping as a Key Element of Sample Size Optimization in Bioequivalence of Risperidone Tablets

Ying Chen, Yang Deng, Miao Yan, Zhenyan Hou, Yao Li, Bikui Zhang, Hualin Cai

Original Research Article

Metabolism of Rhizoma coptidis in Human Urine by Ultra-High-Performance Liquid Chromatography Coupled with High-Resolution Mass Spectrometry

Qingshan Zhang, Gaowa Wang, Xi Chen, Zhiqiang Han, Xiangmei Chen, Risu Na, Haburi Jin, Ping Li, Renbatu Bu

Original Research Article

Prediction of Human Pharmacokinetics of Ulixertinib, a Novel ERK1/2 Inhibitor from Mice, Rats, and Dogs Pharmacokinetics

Ponnayyan Sulochana Suresh, Ravi Kumar Jairam, Devaraj V. Chandrasekhar, Anera Balakrishna Vinod, Rakesh A. Hiremath, Anusha Raj, Mohd Zainuddin, Ravi Kanth Bhamidipati, Ramesh Mullangi

Open Access Original Research Article

Population Pharmacokinetic Analysis and Model-Based Simulations of Aripiprazole for a 1-Day Initiation Regimen for the Long-Acting Antipsychotic Aripiprazole Lauroxil

Marjie L. Hard, Angela Y. Wehr, Brian M. Sadler, Richard J. Mills, Lisa von Moltke