Skip to main content

European Journal of Drug Metabolism and Pharmacokinetics

Ausgabe 5/2016

Inhalt (19 Artikel)

Review Article

Clinical Drug–Drug Pharmacokinetic Interaction Potential of Sucralfate with Other Drugs: Review and Perspectives

Suresh P. Sulochana, Muzeeb Syed, Devaraj V. Chandrasekar, Ramesh Mullangi, Nuggehally R. Srinivas

Original Research Article

Impact of the Cytochrome P450 2B6 (CYP2B6) Gene Polymorphism c.516G>T (rs3745274) on Propofol Dose Variability

Artemísia L. Mourão, Fabiana G. de Abreu, Marilu Fiegenbaum

Original Research Article

Formulation and Pharmacokinetic Evaluation of Polymeric Dispersions Containing Valsartan

Naveen Chella, Bhaskar Daravath, Dinesh Kumar, Rama Rao Tadikonda

Original Paper

Population Pharmacokinetic Analysis of the Oral Absorption Process and Explaining Intra-Subject Variability in Plasma Exposures of Imatinib in Healthy Volunteers

Ali-Akbar Golabchifar, Saeed Rezaee, Nahid Mobarghei Dinan, Abbas Kebriaeezadeh, Mohammad-Reza Rouini

Original Research Article

Pharmacokinetics and Tolerability of Rufinamide Following Single and Multiple Oral Doses and Effect of Food on Pharmacokinetics in Healthy Chinese Subjects

Mingzhen Xu, Yang Ni, Ying Zhou, Xiaomeng He, Huqun Li, Hui Chen, Weiyong Li

Original Paper

Drug–Drug Interactions of a Novel κ-Opioid Receptor Agonist, Nalfurafine Hydrochloride, Involving the P-Glycoprotein

Akihiro Ando, Shinichiro Sasago, Yoshihiro Ohzone, Yohei Miyamoto

Original Paper

Gender-Related Differences in the Expression of Organic Cation Transporter 2 and its Role in Urinary Excretion of Metformin in Rats

Yan-rong Ma, Hong-yan Qin, Yong-wen Jin, Jing Huang, Miao Han, Xing-dong Wang, Guo-qiang Zhang, Yan Zhou, Zhi Rao, Xin-an Wu

Original Paper

Pharmacokinetics of IDX184, a liver-targeted oral prodrug of 2′-methylguanosine-5′-monophosphate, in the monkey and formulation optimization for human exposure

Xin-Ru Pan-Zhou, Benjamin A. Mayes, Hassan Rashidzadeh, Rahela Gasparac, Steven Smith, Sanjeev Bhadresa, Kusum Gupta, Marita Larsson Cohen, Charlie Bu, Steven S. Good, Adel Moussa, Roger Rush

Original Paper

Combining Chemical Permeation Enhancers for Synergistic Effects

Trizel du Toit, Maides M. Malan, Hendrik J. R. Lemmer, Chrisna Gouws, Marique E. Aucamp, Wilma J. Breytenbach, Josias H. Hamman

Original Paper

The Pharmacokinetics and Tissue Distribution of Honokiol and its Metabolites in Rats

Wang Jun-jun, Miao Xiao-lei, Chen Jing-ya, Chen Yong

Original Paper

A Method of Effectively Improved α-Mangostin Bioavailability

Yan Zhao, Guosheng Tang, Qiang Tang, Jing Zhang, Yingying Hou, Enbo Cai, Shuangli Liu, Daihong Lei, Lianxue Zhang, Shijie Wang

Original Paper

Chronopharmacokinetics of Erlotinib and Circadian Rhythms of Related Metabolic Enzymes in Lewis Tumor-Bearing Mice

Jiao Liu, Chun-Yan Wang, Song-Gang Ji, Xia Xu, Pei-Pei Wang, Bin Zhang, Li-Yan Zhao, Liang Liu, Ping-Ping Lin, Le-Kun Liu, Ming-Chun Li

Short Communication

Increased Intestinal Absorption of Genistein by Coadministering Verapamil in Rats

Baogang Xie, Huiyun Wang, Huiqin Zou, Yalan Liu, Xiangyu Kong, Xiuzhong Fang

Short Communication

Microbial Metabolism of Atovaquone and Cytotoxicity of the Produced Phase I Metabolite

Eliane de Oliveira Silva, Natália dos Santos Gonçalves, Raquel Alves dos Santos, Niege Araçari Jacometti Cardoso Furtado

Erratum

Erratum to: Effect of Aroma and Magnum Hops Extracts and Paracetamol on Antioxidant Liver Parameters in Mice

Vida Jakovljevic, Mira Popovic, Aleksandar Raskovic, Ana Sabo, Olga Horvat, Radoslav Mitic, Radica Vasic

Erratum

Erratum to: Interaction of Alcoholic Extracts of Hops with Pentobarbital and Diazepam in Mice

Aleksandar Raskovic, Olga Horvat, Vida Jakovljevic, Jan Sabo, Radica Vasic